Resultados de búsqueda - Drugs Drugs

  1. Targeting Leishmania infantum Mannosyl-oligosaccharide glucosidase with natural products : potential pH-dependent inhibition explored through computer-aided drug design por Goyzueta-Mamani, Luis Daniel, Barazorda-Ccahuana, Haruna Luz, Candia-Puma, Mayron Antonio, Galdino, Alexsandro Sobreira, Machado-de-Avila, Ricardo Andrez, Giunchetti, Rodolfo Cordeiro, Medina-Franco, José L., Florin-Christensen, Mónica, Ferraz Coelho, Eduardo Antonio, Chavez Fumagalli, Miguel Angel

    Publicado 2024
    “…Using computer-aided drug design (CADD) approaches, the potential inhibitory effect of these NP candidates was evaluated by inhibiting the Mannosyl-oligosaccharide Glucosidase Protein (MOGS) from Leishmania infantum, an enzyme essential for the protein glycosylation process, at various pH to mimic the parasite’s changing environment. …”
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  2. Structure-based drug design for envelope protein E2 uncovers a new class of bovine viral diarrhea inhibitors that block virus entry por Pascual, María José, Merwaiss, Fernando, Leal, Emilse Soledad, Quintana, Maria Eugenia, Capozzo, Alejandra Victoria, Cavasotto, Claudio Norberto, Bollini, Mariela, Alvarez, Diego Ezequiel

    Publicado 2019
    “…Using reverse genetics we constructed a recombinant BVDV expressing GFP that served as a sensitive reporter for the study of the mechanism of action of antiviral compounds. Time of drug addition assays showed that PTC12 inhibited an early step of infection. …”
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